- concentration) Rat
DATTooltip Dopamine transporter 29,000 (IC50) Rat
VDCCTooltip Voltage-dependent
calcium channel >10,000 Rat
Values are Ki (nM), unless...
- 220–3,651 >10,000 ND σ2 1,344 1,050 ND NMDA (PCP) >10,000 ND
Antagonist VDCCTooltip Voltage-dependent
calcium channel >10,000 ND ND
hERGTooltip Human Ether-à-go-go-Related...
- 10000+ 10000+ (IC50) 6310 (pA2) 3800
Human Mouse Rat
Guinea pig
Bovine VDCCTooltip Voltage-dependent
calcium channel 3400+ (IC50) Rat
Values are Ki (nM)...
-
receptor 670
Human VGSCTooltip Voltage-gated
sodium channel 6905 Rat
VDCCTooltip Voltage-dependent
calcium channel 10000+ Rat
Values are Ki (nM). The...
-
nAChTooltip Nicotinic acetylcholine receptor 10000+ ND NMDA (PCP) 10000+ ND
VDCCTooltip Voltage-dependent
calcium channel 10000+ ND
VGSCTooltip Voltage-gated...
-
nAChTooltip Nicotinic acetylcholine receptor >10,000 ND NMDA (PCP) >10,000 ND
VDCCTooltip Voltage-dependent
calcium channel >10,000 ND
VGSCTooltip Voltage-gated...
- 000
Guinea pig σ2 >10,000 Rat I1 >10,000
Human A1 >10,000 (EC50)
Human VDCCTooltip Voltage-dependent
calcium channel >10,000
Human Values are Ki (nM), unless...
-
acetylcholine receptors >10,000
Human σ1 ND ND ND σ2 8,350 Rat I1 759 Rat
VDCCTooltip Voltage-dependent
calcium channel 6,043 Rat
Values are Ki (nM). The smaller...
