- directly, a
corresponding prodrug can be used to
improve how the drug is absorbed, distributed, metabolized, and
excreted (ADME).
Prodrugs are
often designed...
- Hypoxia-activated
prodrugs are
prodrugs that
target regions of
tumor hypoxia within tumor cells.
These types of
drugs have the potential,
alone and in...
- medicine,
neurotransmitter prodrugs have also been used as
recreational drugs in some cases.
Monoamine neurotransmitter prodrugs include the catecholamine...
- and
includes the
following marketed medications:
Several of
these act as
prodrugs of norethisterone,
including norethisterone acetate,
norethisterone enanthate...
- This is a list of androgens/anabolic
steroids (AAS) or
testosterone derivatives.
Androgen esters are
mostly not
included in this list. The
major classes...
-
Directed enzyme prodrug therapy (DEPT) uses
enzymes artificially introduced into the body to
convert prodrugs,
which have no or poor
biologically activity...
- levodopa/carbidopa/entacapone). In
addition to
levodopa itself,
certain prodrugs of
levodopa are available,
including melevodopa (melevodopa/carbidopa)...
- 30 minutes and did not
differ between 4-AcO-DMT and psilocybin.
Psilocin ester prodrugs like 4-AcO-DMT are
cleaved into
psilocin by
esterase enzymes. A 2025 in...
-
prepare ester prodrugs which have
increased half-lives
relative to the
parent compound. The
lipophilicity of the
cypionate group allows the
prodrug to be sequestered...
- of mometasone, is the
marketed medication.
Mometasone furoate acts as a
prodrug of mometasone. In
addition to its
glucocorticoid activity,
mometasone also...
