- directly, a
corresponding prodrug can be used to
improve how the drug is absorbed, distributed, metabolized, and
excreted (ADME).
Prodrugs are
often designed...
- medicine,
neurotransmitter prodrugs have also been used as
recreational drugs in some cases.
Monoamine neurotransmitter prodrugs include the catecholamine...
- and
includes the
following marketed medications:
Several of
these act as
prodrugs of norethisterone,
including norethisterone acetate,
norethisterone enanthate...
- Hypoxia-Activated
Prodrugs (HAPs) are
prodrugs that
target regions of
tumor hypoxia within tumor cells. HAPs may
offer the potential,
alone and in combination...
- levodopa/carbidopa/entacapone). In
addition to
levodopa itself,
certain prodrugs of
levodopa are available,
including melevodopa (melevodopa/carbidopa)...
- This is a list of androgens/anabolic
steroids (AAS) or
testosterone derivatives.
Androgen esters are
mostly not
included in this list. The
major classes...
- use are rash and
gastrointestinal upset,
including nausea and vomiting.
Prodrugs that
release pivalate anions when
broken down by the body — such as pivmecillinam...
- His main
research focus has been on the
design and
characterization of
prodrugs and
protoxins targeted for
activation by
cancer specific proteases. This...
-
called prodrugs. The
reasons for this type of
formulation may be
because the drug is more
stable during manufacture and
storage as the
prodrug form, or...
-
Directed enzyme prodrug therapy (DEPT) uses
enzymes artificially introduced into the body to
convert prodrugs,
which have no or poor
biologically activity...
