- A
prodrug is a
pharmacologically inactive medication or
compound that,
after intake, is
metabolized (i.e.,
converted within the body) into a pharmacologically...
-
neurotransmitter prodrug, or
neurotransmitter precursor, is a drug that acts as a
prodrug of a neurotransmitter. A
variety of
neurotransmitter prodrugs have been...
- research. However,
norethisterone enanthate, an
intramuscularly administered prodrug of
norethisterone which is used as a long-acting contraceptive, is used...
-
Directed enzyme prodrug therapy (DEPT) uses
enzymes artificially introduced into the body to
convert prodrugs,
which have no or poor
biologically activity...
- (γ-hydroxybutyric acid acetate) –
synthetic prodrug to GHB GBL (γ-hydroxybutyric acid lactone) –
metabolic intermediate and
prodrug to GHB
GHBAL (γ-hydroxybutyraldehyde...
-
benzodiazepine receptor) than the
benzodiazepine receptor.
Gidazepam acts as a
prodrug to its
active metabolite 7-bromo-2,3-dihydro-5-phenyl-1H-1,4-benzodiazepin-2-one...
- Hypoxia-Activated
Prodrugs (HAPs) are
prodrugs that
target regions of
tumor hypoxia within tumor cells. HAPs may
offer the potential,
alone and in combination...
-
psilocybin for
pharmacological studies, as they are both
believed to be
prodrugs of psilocin. However, some
users report that O-acetylpsilocin's subjective...
-
called prodrugs. The
reasons for this type of
formulation may be
because the drug is more
stable during manufacture and
storage as the
prodrug form, or...
-
derivative which is
thought to act as a
prodrug for DOC and
theophylline in the same way in
which fenethylline acts as a
prodrug for
amphetamine and theophylline...