- A
prodrug is a
pharmacologically inactive medication or
compound that,
after intake, is
metabolized (i.e.,
converted within the body) into a pharmacologically...
-
Directed enzyme prodrug therapy (DEPT) uses
enzymes artificially introduced into the body to
convert prodrugs,
which have no or poor
biologically activity...
- research. However,
norethisterone enanthate, an
intramuscularly administered prodrug of
norethisterone which is used as a long-acting contraceptive, is used...
- with an
acetate ester. The drug is a
prodrug of
psilocin and is
orally active similarly to psilocybin. As a
prodrug of psilocin, 4-AcO-DMT acts as a non-selective...
-
neurotransmitter prodrug, or
neurotransmitter precursor, is a drug that acts as a
prodrug of a neurotransmitter. A
variety of
neurotransmitter prodrugs have been...
-
psychedelic of the
tryptamine family. It acts as a
prodrug of
psilocin (4-HO-DMT)
similarly to
other psilocin prodrugs like 4-AcO-DMT, 4-PrO-DMT, and psilocybin...
- Hypoxia-activated
prodrugs are
prodrugs that
target regions of
tumor hypoxia within tumor cells.
These types of
drugs have the potential,
alone and in...
- of mometasone, is the
marketed medication.
Mometasone furoate acts as a
prodrug of mometasone. In
addition to its
glucocorticoid activity,
mometasone also...
-
among others. The drug is a
centrally permeable monoamine precursor and
prodrug of
dopamine and
hence acts as a
dopamine receptor agonist. Chemically,...
-
Alprazolam triazolobenzophenone is a
chemical compound that is a
prodrug for the
benzodiazepine derivative alprazolam. At
neutral pH it
readily cyclizes...