-
Piromelatine (Neu-P11) is a
multimodal sleep drug
under development by
Neurim Pharmaceuticals. It is an
agonist at
melatonin MT1/MT2 and
serotonin 5-HT1A/5-HT1D...
- (N-acetylserotonin; NAS) N-Acetyltryptamine N-Butanoylmelatonin N-Propionylmelatonin
Piromelatine TIK-301 (LY-156735) α-Alkyltryptamines 1-Methyl-AMT 2,α-DMT (2-Me-AMT)...
-
results of a
positive phase II
trial of its
investigational compound piromelatine (Neu-P11) in
February 2013. No
antagonists or
selective ligands are currently...
- (N-acetylserotonin; NAS) N-Acetyltryptamine N-Butanoylmelatonin N-Propionylmelatonin
Piromelatine TIK-301 (LY-156735) α-Alkyltryptamines 1-Methyl-AMT 2,α-DMT (2-Me-AMT)...
- (N-acetylserotonin; NAS) N-Acetyltryptamine N-Butanoylmelatonin N-Propionylmelatonin
Piromelatine TIK-301 (LY-156735) α-Alkyltryptamines 1-Methyl-AMT 2,α-DMT (2-Me-AMT)...
- (N-acetylserotonin; NAS) N-Acetyltryptamine N-Butanoylmelatonin N-Propionylmelatonin
Piromelatine TIK-301 (LY-156735) α-Alkyltryptamines 1-Methyl-AMT 2,α-DMT (2-Me-AMT)...
-
agonists used in
medicine like ramelteon, tasimelteon, agomelatine, and
piromelatine (still in
clinical trials) are
analogues of melatonin. The
first patent...
-
Fabomotizole (afobazole) GR-196,429
Melatonin N-Acetylserotonin (normelatonin)
Piromelatine Ramelteon Tasimelteon TIK-301 (LY-156,735) Antagonists:
Luzindole MT2Tooltip...
- (N-acetylserotonin; NAS) N-Acetyltryptamine N-Butanoylmelatonin N-Propionylmelatonin
Piromelatine TIK-301 (LY-156735) α-Alkyltryptamines 1-Methyl-AMT 2,α-DMT (2-Me-AMT)...
- (N-acetylserotonin; NAS) N-Acetyltryptamine N-Butanoylmelatonin N-Propionylmelatonin
Piromelatine TIK-301 (LY-156735) α-Alkyltryptamines 1-Methyl-AMT 2,α-DMT (2-Me-AMT)...