- group, such as an azide, a
diazirine or a benzophenone.
Photoaffinity labeling Photoaffinity labeling, Gold Book Ruoho, A. E.; Kiefer, H.; Roeder, P....
- small, photo-reactive,
crosslinking reagents. They are
often used in
photoaffinity labeling studies to
observe a
variety of interactions,
including ligand-receptor...
-
residues in the
receptor and
become covalently bound to the receptor.
Photoaffinity labeling "Pharmacology of cell excitation".
Biochemical Pharmacology...
-
Unlike ABPP,
which results in
protein labeling upon
probe binding,
photoaffinity labeling probes require activation by
photolysis before covalent bonding...
- photoreactions,
isoxazole group is
developed as a
native photo-cross-linker for
photoaffinity labeling and
chemoproteomic studies.
Isoxazoles also form the basis...
- Pichler, G; Holdt, LM; Teupser, D; Mann, M;
Chuang (November 2013). "
Photoaffinity labeling of
plasma proteins". Molecules. 18 (11): 13831–13859. doi:10...
-
research charity (N,N-dimethyl-amino)-benzenediazonium-fluoroborate, a
photoaffinity probe that
competes with
acetylcholine for
receptor binding Sulfoxone...
-
ligand in
androgen receptor (AR)
ligand binding ****ays (LBAs) and as a
photoaffinity label for the AR. More precisely,
metribolone is the 17α-methylated...
- antagonist.
Niznik HB, Guan JH,
Neumeyer JL,
Seeman P (February 1985). "A
photoaffinity ligand for
dopamine D2 receptors: azidoclebopride".
Molecular Pharmacology...
-
literature has
commenced on the
requirement of off-pathway catalysis.
Photoaffinity labels are
characterized by
nonenzymatic reactivity produced by exposure...