-
unambiguously denotes molar. Sub-multiples, such as "millimolar" (mM) and "
nanomolar" (nM),
consist of the unit
preceded by an SI prefix: The
conversion to...
- Ether-à-go-go-Related Gene 34,000–69,000 IC50
Human Notes: (1)
Values are in
nanomolar (nM) units. The
smaller the value, the more
avidly the drug
binds to or...
- accordance,
while gabapentinoids like
pregabalin and
gabapentin have
nanomolar affinities for the α2δ subunit,
their potencies in vivo are in the low...
- seven, four of
which are
highly expressed in the
human brain, with low
nanomolar through low
micromolar activating effects.
Based upon
preclinical research...
-
purification of that
class of ion
channels and gave its name to it. At
nanomolar concentrations,
ryanodine locks the
receptor in a half-open state, whereas...
-
Neurotransmitter transporter Measure (units) dl-MPH d-MPH l-MPH DAT Ki (nMTooltip
nanomolar) 121 161 2250 IC50 (nM) 20 23 1600 NET Ki (nM) 788 206 >10000 IC50 (nM)...
-
antagonize the
effects of gabapentin. Accordingly,
while gabapentin has
nanomolar affinity for the α2δ subunit, its
potency in vivo is in the low micromolar...
-
together with
ziprasidones also weak
nanoMolar ability of 112)
brexpiprazole has just the weak DAT-transporter
nanoMolar affinity of the
multiple of 0.8 compared...
- CM156 is a
piperazine based chemical compound with
nanomolar affinity for both
sigma receptor subtypes that has been
shown to
counteract the deleterious...
-
competitively binding to both wild-type and
mutant estrogen receptors with
nanomolar potency.
Giredestrant works by
inducing an
inactive conformation of the...
