-
unambiguously denotes molar. Sub-multiples, such as "millimolar" (mM) and "
nanomolar" (nM),
consist of the unit
preceded by an SI prefix: The
conversion to...
- Ether-à-go-go-Related Gene 34,000–69,000 IC50
Human Notes: (1)
Values are in
nanomolar (nM) units. The
smaller the value, the more
avidly the drug
binds to or...
-
Neurotransmitter transporter Measure (units) dl-MPH d-MPH l-MPH DAT Ki (nMTooltip
nanomolar) 121 161 2250 IC50 (nM) 20 23 1600 NET Ki (nM) 788 206 >10000 IC50 (nM)...
- Methaemoglobinaemia*
Metoclopramide appears to bind to
dopamine D2
receptors with
nanomolar affinity (Ki = 28.8 nM),
where it is a
receptor antagonist, and is also...
-
antagonize the
effects of gabapentin. Accordingly,
while gabapentin has
nanomolar affinity for the α2δ subunit, its
potency in vivo is in the low micromolar...
- seven, four of
which are
highly expressed in the
human brain, with low
nanomolar through low
micromolar activating effects.
Based upon
preclinical research...
-
receptor 1, with
picomolar binding affinity, and
melatonin receptor 2, with
nanomolar binding affinity. Both
receptors are part of the G-protein
coupled receptors...
- accordance,
while gabapentinoids like
pregabalin and
gabapentin have
nanomolar affinities for the α2δ subunit,
their potencies in vivo are in the low...
-
acting growth factors.
classic hormones circulate in
aqueous solution in
nanomolar (10-9 M)
concentrations that
usually vary by less than one
order of magnitude...
-
adrenergic receptors as well as the
histamine H1 receptor. It has sub-
nanomolar affinity for the
dopamine D2, and D3 receptors,
serotonin 5-HT1A and 5-HT1D...
