- 6β-
Naltrexol, or 6β-hydroxynaltrexone (developmental code name AIKO-150), is a peripherally-selective
opioid receptor antagonist related to naltrexone...
-
concentrations of
naltrexone and 6β-
naltrexol (metabolite) is
within 1 hour.
Linear increases in
circulating naltrexone and 6β-
naltrexol concentrations occur over...
- 6β-
Naltrexol-d4, also
known as 6β-hydroxynaltrexone-d4, is a deuterium-labeled form of 6β-
naltrexol used for NMR imaging.
Unlike opioid inverse agonists...
- 4-Caffeoyl-1,5-quinide 5'-Guanidinonaltrindole β-Funaltrexamine 6β-
Naltrexol 6β-
Naltrexol-d4
Alvimopan AT-076
Binaltorphimine BU09059
Buprenorphine Chlornaltrexamine...
-
remained an off-label option.
Naltrexone and its
active metabolite 6-β-
naltrexol are
competitive antagonists at μ-opioid and κ-opioid receptors, and to...
- 4-Caffeoyl-1,5-quinide 4′-Hydroxyflavanone 4',7-Dihydroxyflavone 6β-
Naltrexol 6β-
Naltrexol-d4 18-MC α-Gliadin β-Chlornaltrexamine β-Funaltrexamine Akuammine...
-
actually be very weak
partial agonists rather than
silent antagonists. 6β-
Naltrexol Alvimopan Axelopran Bevenopran Methylnaltrexone Naldemedine Naloxegol...
- β-Naltrexamine, or 6β-naltrexamine, is an
opioid receptor antagonist related to
naltrexol and naltrexone. It has
served as a
parent pharmacop**** for irreversible...
-
within the
central nervous system.
Alvimopan Methylnaltrexone Naloxegol 6β-
Naltrexol Axelopran Bevenopran Methylsamidorphan Naldemedine Buprenorphine and dezocine...
- 4-Caffeoyl-1,5-quinide 4′-Hydroxyflavanone 4',7-Dihydroxyflavone 6β-
Naltrexol 6β-
Naltrexol-d4 18-MC α-Gliadin β-Chlornaltrexamine β-Funaltrexamine Akuammine...
