-
targets (with Ki
below 100 μM) Site
Value (μM) Type
Action Species Ref
NMDATooltip N-Methyl-D-aspartate
receptor 0.25–0.66 Ki
Antagonist Human MORTooltip...
-
Phencyclidine Site Ki (nM)
Action Species Ref
NMDATooltip N-Methyl-D-aspartate
receptor 59
Antagonist Human MORTooltip μ-Opioid
receptor >10,000 ND Human...
- 5-HT3 2,600 >100,000 σ1 2,500–9,000 11,000–15,000 σ2 90–400 5,000–19,000
NMDATooltip N-Methyl-D-aspartate
receptor 1,000–3,000 6,000–15,000
nAChTooltip Nicotinic...
-
Partial agonist Human 50±10 (8mg≥) σ1 >100,000 ND ND σ2 ND ND ND ND
NMDATooltip N-Methyl-D-aspartate
receptor ND ND ND ND TLR4Tooltip Toll-like receptor...