- (HNK) IC50 NAM Rat ERαTooltip
Estrogen receptor alpha 0.34 Ki ND
Human NETTooltip Norepinephrine transporter 82–291 IC50
Inhibitor Human DATTooltip Dopamine...
- concentration) 50–72 (EC50Tooltip Half-maximal
effective concentration) (rat)
NETTooltip Norepinephrine transporter 27,000–30,500 (Ki) 360–405 (IC50) 54–110 (EC50)...
-
DATTooltip Dopamine transporter (DRIsTooltip
Dopamine reuptake inhibitors)
NETTooltip Norepinephrine transporter (NRIsTooltip
Norepinephrine reuptake inhibitors)...
- 000 (Ki) >100,000 (IC50Tooltip half-maximal
inhibitory concentration)
NETTooltip Norepinephrine transporter 5,600–>30,000 (Ki) >100,000 (IC50) DATTooltip...
-
DATTooltip Dopamine transporter (DRIsTooltip
Dopamine reuptake inhibitors)
NETTooltip Norepinephrine transporter (NRIsTooltip
Norepinephrine reuptake inhibitors)...
- (nM)
Species References SERTTooltip Serotonin transporter 0.15–3.3
Human NETTooltip Norepinephrine transporter 420–925
Human DATTooltip Dopamine transporter...
- Site Ki (nM)
Species Ref
SERTTooltip Serotonin transporter 15.2
Human NETTooltip Norepinephrine transporter 1,440
Human DATTooltip Dopamine transporter...
-
DATTooltip Dopamine transporter (DRIsTooltip
Dopamine reuptake inhibitors)
NETTooltip Norepinephrine transporter (NRIsTooltip
Norepinephrine reuptake inhibitors)...
-
Clonidine Site Ki (nM)
Species Ref
NETTooltip Norepinephrine transporter >1,000
Human 5-HT1B >10,000 Rat 5-HT2A >10,000
Human α1A 316.23
Human α1B 316...
- MK-801/PCPTooltip
phencyclidine site
SERTTooltip Serotonin transporter and
NETTooltip norepinephrine transporter blocker (cf. serotonin–norepinephrine reuptake...
