- concentration) 50–72 (EC50Tooltip Half-maximal
effective concentration) (rat)
NETTooltip Norepinephrine transporter 27,000–30,500 (Ki) 360–405 (IC50) 54–110 (EC50)...
- MK-801/PCPTooltip
phencyclidine site
SERTTooltip Serotonin transporter and
NETTooltip norepinephrine transporter blocker (cf. serotonin–norepinephrine reuptake...
-
DATTooltip Dopamine transporter (DRIsTooltip
Dopamine reuptake inhibitors)
NETTooltip Norepinephrine transporter (NRIsTooltip
Norepinephrine reuptake inhibitors)...
- (SERTTooltip
serotonin transporter,
DATTooltip dopamine transporter,
NETTooltip norepinephrine transporter). It is ****ociated with
monoamine reuptake...
- 000 (Ki) >100,000 (IC50Tooltip half-maximal
inhibitory concentration)
NETTooltip Norepinephrine transporter 5,600–>30,000 (Ki) >100,000 (IC50) DATTooltip...
- Site CBP NCBP
Action SERTTooltip Serotonin transporter 108 ND
Inhibitor NETTooltip Norepinephrine transporter 36 ND
Inhibitor DATTooltip Dopamine transporter...
- 100 (IC50Tooltip Half-maximal
inhibitory concentration) 81–114 (EC50)
NETTooltip Norepinephrine transporter 6,500–>10,000 (Ki) 3,900 (IC50) 4,166 (EC50)...
-
DATTooltip Dopamine transporter (DRIsTooltip
Dopamine reuptake inhibitors)
NETTooltip Norepinephrine transporter (NRIsTooltip
Norepinephrine reuptake inhibitors)...
- (IC50Tooltip half-maximal
inhibitory concentration) 561 (EC50) 54% (Emax)
NETTooltip Norepinephrine transporter 13,000 (Ki) 14,000 (IC50) >10,000 (EC50) DATTooltip...
- (HNK) IC50 NAM Rat ERαTooltip
Estrogen receptor alpha 0.34 Ki ND
Human NETTooltip Norepinephrine transporter 82–291 IC50
Inhibitor Human DATTooltip Dopamine...