-
Mepyramine, also
known as pyrilamine, is a first-generation antihistamine,
targeting the H1
receptor as an
inverse agonist.
Mepyramine rapidly permeates...
- that of atropine,
while its
antihistamine activity approaches that of
mepyramine. Its
anticholinergic effects have been
established as therapeutically...
-
discovered in 1933 at the
Pasteur Institute in France, and also
including mepyramine, tripelennamine, and antazoline. The
other classes are
derivatives of...
- "Histamine H1
receptors identified in
mammalian brain membranes with [3H]
mepyramine".
Proceedings of the
National Academy of
Sciences of the
United States...
- S,
Young JM (November 1995). "Characteristics of the
binding of [3H]-
mepyramine to
intact human U373 MG
astrocytoma cells:
evidence for histamine-induced...
-
Dextropropoxyphene (Darvon)
Dimenhydrinate (Dramamine)
Diphenhydramine (Benadryl)
Mepyramine (pyrilamine) (Anthisan)
Mifepristone (Korlym, Mifeprex) 4′-Fluorococaine...
- g., brompheniramine, chlorphenamine, dimenhydrinate, diphenhydramine,
mepyramine (pyrilamine), pheniramine, tripelennamine)
Antipsychotics (e.g., loxapine...
- EA-3443 EA-3580 EA-3834
Flavoxate Hyoscyamine JB-318 JB-336
Meclozine Mepyramine Orphenadrine Oxybutynin Pheniramine Phenyltoloxamine Procyclidine Promethazine...
- g., brompheniramine, chlorphenamine, dimenhydrinate, diphenhydramine,
mepyramine (pyrilamine), pheniramine, tripelennamine)
Antipsychotics (e.g., loxapine...
-
Hydroxyethylpromethazine Hydroxyzine Isopromethazine Isothipendyl Meclozine Medrylamine Mepyramine (pyrilamine)
Mequitazine Methafurylene Methapyrilene Methdilazine Moxastine...
