- 2]-cycloaddition of
nitrile oxides and 1,3-****tones, β-ketoesters, or β-
ketoamides".
Beilstein J. Org. Chem. (18): 446–458. doi:10.3762/bjoc.18.47. PMC 9039522...
-
Intermolecular Hydroacylation:
Enantioselective Cross-Coupling of
Aldehydes and
Ketoamides".
Journal of the
American Chemical Society. 136 (26): 9471–9476. doi:10...
- "Direct and
Highly Enantioselective Iso-Pictet-Spengler
Reactions with α-
Ketoamides:
Access to
Underexplored Indole Core Structures". Org. Lett. 14 (10):...
- copper-catalyzed
catalytic enantioselective Mannich reaction using 2H-azirines and β-
ketoamides. The
racemic 2H-azirines was
first applied and one
enantiomer of the 2H-azirine...
-
carbamate derivatized norleucine aldehyde 1tu6:
Cathepsin K
complexed with a
ketoamide inhibitor 1u9v:
Crystal Structure of the
Cysteine Protease Human Cathepsin...
-
formation of
structures like α-amino acids, α-hydroxy-β-amino acids, α-
ketoamides, β-
ketoamides, α-hydroxyketones and α-aminoxyamides. The P****erini
reaction has...
-
Zhang L, Lin D,
Kusov Y, Nian Y, Ma Q, Wang J, et al. (February 2020). "α-
Ketoamides as Broad-Spectrum
Inhibitors of
Coronavirus and
Enterovirus Replication:...
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Regner F,
Vierling M, Möller A (June 2003). "Benzoylalanine-derived
ketoamides carrying vinylbenzyl amino residues:
discovery of
potent water-soluble...
- of SARS-CoV-2 main
protease provides a
basis for
design of
improved α-
ketoamide inhibitors". Science. 368 (6489): 409–412. Bibcode:2020Sci...368..409Z...
- of the side-chain
followed by Wipf and Miller's
cyclodehydration of β-
ketoamides described above.
Lilly Research Laboratories has
disclosed the structure...
