-
Ketanserin, sold
under the
brand name Sufrexal, is an
antihypertensive agent which is used to
treat arterial hypertension and
vasospastic disorders. It...
- than
ketanserin at
blocking psilocybin's effects, but risperidone, an
antipsychotic with
combined D2/5-HT2 activity, is as
effective as
ketanserin (Vollenweider...
- psychedelics. Accordingly, the
serotonin 5-HT2A
receptor antagonists ketanserin, an
antihypertensive agent, and risperidone, an antipsychotic, have been...
-
derived by
structural modification of the
selective 5-HT2A
antagonist ketanserin, with the 4-(p-fluorobenzoyl)piperidine
moiety replaced by the N-(2-methoxybenzyl)...
-
receptor antagonist GR-55562 and the
serotonin 5-HT2A
receptor antagonist ketanserin were both ineffective. Likewise,
another study found that
selective antagonists...
- (Atarax) (minor effect)
Ketanserin – The
discovery of
ketanserin was a
landmark in the
pharmacology of 5-HT2 receptors.
Ketanserin,
though capable of blocking...
-
effects of the
lysergic acid
diethylamide (LSD) in animals, and,
along with
ketanserin, led to the
elucidation of the 5-HT2A
receptor as the
biological mediator...
-
dopamine receptors D1 and D2,
histamine receptor H1, and A1 adrenoreceptors.
Ketanserin Antihypertensive.
Blocks 5-HT2A, 5-HT2C and
Alpha 1 (A1) adrenoreceptors...
- Deutetrabe****ne Dihydrotetrabe****ne
Efavirenz GBR-12935 GZ-793A
Ibogaine Ketanserin Lobeline Methoxytetrabe****ne
Reserpine Rose
bengal Tetrabe****ne Valbe****ne...
-
serotonergic psychedelics.
Serotonin 5-HT2A
receptor antagonists like
ketanserin and
risperidone have been
found to
fully block or dose-dependently reduce...
