-
Kainate receptors, or
kainic acid
receptors (KARs), are
ionotropic receptors that
respond to the
neurotransmitter glutamate. They were
first identified...
-
Kainic acid, or
kainate, is an acid that
naturally occurs in some seaweed.
Kainic acid is a
potent neuroexcitatory amino acid
agonist that acts by activating...
- receptors: AMPA and
kainate receptors.
Willardiine analogs have been
developed that have
different binding affinities for the AMPA and
kainate receptors. These...
- receptors, and
metabotropic glutamate receptors. A
fourth class,
known as
kainate receptors, are
similar in many
respects to AMPA receptors, but much less...
-
cyanquixaline (6-cyano-7-nitroquinoxaline-2,3-dione) is a
competitive AMPA/
kainate receptor antagonist. Its
chemical formula is C9H4N4O4. CNQX is
often used...
-
Glutamate receptor, ionotropic,
kainate 1, also
known as GRIK1, is a
protein that in
humans is
encoded by the GRIK1 gene. This gene
encodes one of the...
- a
selective agonist for the
kainate receptor, with only
limited effects at the AMPA receptor. It is
selective for
kainate receptors composed of GluR5...
-
damaged neurons.
Riluzole has also been
reported to
directly inhibit the
kainate and NMDA receptors. The drug has also been
shown to
postsynaptically potentiate...
- of the AMPA and
kainate subtypes of the
ionotropic glutamate receptor family, with
selectivity for the GluR5
subtype of the
kainate receptor. It has...
-
selective agonist for the
kainate receptor. This
potent agonist has
nearly 3,000 fold- and 200-fold
selectivity for
kainate receptors over AMPA and NMDA...
