- are known, 2-
imidazolines, 3-
imidazolines, and 4-
imidazolines. The 2- and 3-
imidazolines contain an
imine center,
whereas the 4-
imidazolines contain an...
-
Imidazoline receptors are the
primary receptors on
which clonidine and
other imidazolines act.
There are
three main
classes of
imidazoline receptor: I1...
-
peripheral vasomotor structures.
Rilmenidine is a
imidazoline analog and
shows greater selectivity for
imidazoline receptors than for
cerebral alpha2-adrenergic...
- 2-
Imidazoline (Preferred
IUPAC name: 4,5-dihydro-1H-imidazole) is one of
three isomers of the nitrogen-containing
heterocycle imidazoline, with the formula...
-
Moxonidine (INN) is a new-generation alpha-2/
imidazoline receptor agonist antihypertensive drug
licensed for the
treatment of mild to
moderate essential...
-
example of autoreceptor. However, it is now
known that
clonidine binds to
imidazoline receptors with a much
greater affinity than α2 receptors,
which would...
-
certain oral
medications (e.g.,
sympathomimetic amines and
various 2-
imidazolines) that
constrict blood vessels in the
lining of the nose,
although evidence...
-
Selected examples are:
Brimonidine Clonidine (mixed alpha2-adrenergic and
imidazoline-I1
receptor agonist)
Dexmedetomidine Fadolmidine Guanfacine, (preference...
-
ingested the drug.
There is no
antidote for
tetryzoline or
other similar imidazoline analogue poisoning, but the
symptoms can be alleviated. With treatment...
- (NAR) up to 35.7% and
reduce nasal mucosal blood flow up to 50%.
Since imidazolines are
sympathomimetic agents,
their primary effects appear on α adrenergic...
