-
Imidazoline receptors are the
primary receptors on
which clonidine and
other imidazolines act.
There are
three main
classes of
imidazoline receptor: I1...
- are known, 2-
imidazolines, 3-
imidazolines, and 4-
imidazolines. The 2- and 3-
imidazolines contain an
imine center,
whereas the 4-
imidazolines contain an...
- 2-
Imidazoline (Preferred
IUPAC name: 4,5-dihydro-1H-imidazole) is one of
three isomers of the nitrogen-containing
heterocycle imidazoline, with the formula...
-
example of autoreceptor. However, it is now
known that
clonidine binds to
imidazoline receptors with a much
greater affinity than α2 receptors,
which would...
- the
presence of para-toluenesulfonic acid to form the
corresponding imidazoline, this
being xylometazoline.
Carbon disulfide can also be used as a catalyst...
-
vascular resistance.: 201–203
Clonidine also acts as an
agonist at
imidazoline-1 (I1)
receptors in the brain, and it is
hypothesized that this effect...
-
selective α2-adrenergic
receptor antagonist, and an
antagonist for the
imidazoline receptor.
Idazoxan has been
under investigation as an antidepressant...
-
Selected examples are:
Brimonidine Clonidine (mixed alpha2-adrenergic and
imidazoline-I1
receptor agonist)
Dexmedetomidine Fadolmidine Guanfacine, (preference...
-
peripheral vasomotor structures.
Rilmenidine is a
imidazoline analog and
shows greater selectivity for
imidazoline receptors than for
cerebral alpha2-adrenergic...
-
Moxonidine (INN) is a new-generation alpha-2/
imidazoline receptor agonist antihypertensive drug
licensed for the
treatment of mild to
moderate essential...
