-
Galeterone (developmental code
names TOK-001, VN/124-1) is a
steroidal antiandrogen which was
under development by
Tokai Pharmaceuticals for the treatment...
- and
prevents mineralocorticoid excess.
Abiraterone acetate,
along with
galeterone, has been
identified as an
inhibitor of
sulfotransferases (SULT2A1, SULT2B1b...
-
known structures while bound to two
steroidal inhibitors,
abiraterone and
galeterone, CYP17A1
possesses the
canonical cytochrome P450 fold
present in other...
- DU-41165
Edogestrone EM-4350 EM-5854 EM-5855 EM-6537
Epitestosterone Galeterone Guggulsterone Ludaterone Medrogestone Megestrol acetate Mespirenone Metogest...
- DU-41165
Edogestrone EM-4350 EM-5854 EM-5855 EM-6537
Epitestosterone Galeterone Guggulsterone Ludaterone Medrogestone Megestrol acetate Mespirenone Metogest...
- DU-41165
Edogestrone EM-4350 EM-5854 EM-5855 EM-6537
Epitestosterone Galeterone Guggulsterone Ludaterone Medrogestone Megestrol acetate Mespirenone Metogest...
- DU-41165
Edogestrone EM-4350 EM-5854 EM-5855 EM-6537
Epitestosterone Galeterone Guggulsterone Ludaterone Medrogestone Megestrol acetate Mespirenone Metogest...
- drug
ketoconazole and the
newer drugs abiraterone acetate, orteronel,
galeterone, and seviteronel. CYP17A1 inhibitors, such as
abiraterone acetate, are...
- DU-41165
Edogestrone EM-4350 EM-5854 EM-5855 EM-6537
Epitestosterone Galeterone Guggulsterone Ludaterone Medrogestone Megestrol acetate Mespirenone Metogest...
- DU-41165
Edogestrone EM-4350 EM-5854 EM-5855 EM-6537
Epitestosterone Galeterone Guggulsterone Ludaterone Medrogestone Megestrol acetate Mespirenone Metogest...