-
Gabazine (SR-95531) is a drug that acts as an
antagonist at
GABAA receptors. It is used in
scientific research and has no role in medicine, as it would...
-
Varenicline WAY-317,538
Convulsants Anatoxin-a
Bicuculline DMCM
Flurothyl Gabazine Pentetrazol Picrotoxin Strychnine Thujone Eugeroics Adrafinil Armodafinil...
-
receptor agonist Gabamide (γ-aminobutanamide) – GABA
receptor agonist Gabazine (SR-95531) –
antagonist of the
GABAA and GHB
receptors GAVA (γ-aminopentanoic...
- to be
markedly more
potent than the
standard GABAA receptor antagonist gabazine. Frølund B,
Ebert B,
Kristiansen U,
Liljefors T, Krogsgaard-L****n P (August...
- piperidine-4-sulfonic acid (partial agonist).
Orthosteric antagonists: bicuculline,
gabazine.
Positive allosteric modulators: abecarnil,
azocarnil (photoswitchable)...
-
Varenicline WAY-317,538
Convulsants Anatoxin-a
Bicuculline DMCM
Flurothyl Gabazine Pentetrazol Picrotoxin Strychnine Thujone Eugeroics Adrafinil Armodafinil...
-
intrathecal administration of
gabazine, a
GABAA antagonist, in
animals receiving continuous infusions of SP into the RVM.
Gabazine treatment completely reversed...
-
Varenicline WAY-317,538
Convulsants Anatoxin-a
Bicuculline DMCM
Flurothyl Gabazine Pentetrazol Picrotoxin Strychnine Thujone Eugeroics Adrafinil Armodafinil...
-
Varenicline WAY-317,538
Convulsants Anatoxin-a
Bicuculline DMCM
Flurothyl Gabazine Pentetrazol Picrotoxin Strychnine Thujone Eugeroics Adrafinil Armodafinil...
-
Varenicline WAY-317,538
Convulsants Anatoxin-a
Bicuculline DMCM
Flurothyl Gabazine Pentetrazol Picrotoxin Strychnine Thujone Eugeroics Adrafinil Armodafinil...