- The
GABAA receptor (
GABAAR) is an
ionotropic receptor and ligand-gated ion channel. Its
endogenous ligand is γ-aminobutyric acid (GABA), the
major inhibitory...
- In pharmacology,
GABAA receptor positive allosteric modulators, also
known as
GABAkines or
GABAA receptor potentiators, are
positive allosteric modulator...
-
receptors (
GABAAR). A
structural isomer of chloralose, β-chloralose (also
called parachloralose in
older literature), is
inactive as a
GABAAR modulator...
- JR (April 2020). "Subtype
Selective γ-Aminobutyric Acid Type A
Receptor (
GABAAR)
Modulators Acting at the
Benzodiazepine Binding Site: An Update". Journal...
- Nonetheless, the
GABAAR gamma subunit is
palmitoylated and the
alpha subunit binds to PIP2. When the
agonist GABA
binds to
GABAAR it
causes a translocation...
-
Racemorphan Salvinorin A
Spiradoline Tifluadom U-50488 U-69,593
Xorphanol GABAAR agonists Gaboxadol (THIP)
Ibotenic acid (Amanita muscaria)
Muscimol (Amanita...
-
Racemorphan Salvinorin A
Spiradoline Tifluadom U-50488 U-69,593
Xorphanol GABAAR agonists Gaboxadol (THIP)
Ibotenic acid (Amanita muscaria)
Muscimol (Amanita...
- Alzheimer's
disease brain cholesterol was
elevated and
GABAAR shifted into GM1 clusters.
During GABAAR activation by the
neurotransmitter GABA, the receptors...
- Abrepota, Bakeja,
Bharchoondh Bahawalani, Damro, Damhio, Dandio, Detho, Gābar,
Gābaar, Gābhar, Gābrio, Gaad, Gohata, Gandhai, Husrani, Tayuja, Tar'ra, Tanak,...
-
Racemorphan Salvinorin A
Spiradoline Tifluadom U-50488 U-69,593
Xorphanol GABAAR agonists Gaboxadol (THIP)
Ibotenic acid (Amanita muscaria)
Muscimol (Amanita...
