-
Ethisterone, also
known as ethinyltestosterone, pregneninolone, and
anhydrohydroxyprogesterone and
formerly sold
under the
brand names Proluton C and...
- 17α-Ethynylated/vinylated
testosterone derivatives:
ethynyltestosterone (
ethisterone) and
vinyltestosterone derivatives The last
group consists of progestins...
-
parent compounds, testosterone,
nandrolone (19-nortestosterone), and
ethisterone (17α-ethynyltestosterone), have 2%, 22%, and 44% of the
relative binding...
-
affinity and
efficacy of
danazol itself at the PR are
relatively low,
ethisterone, one of the
major metabolites of danazol, is
described as a weak progestogen...
- was
first introduced for
medical use in 1934 and the
first progestin,
ethisterone, was
introduced for
medical use in 1939. More
potent progestins, such...
-
metabolite of the
formerly clinically used but now-discontinued
progestin ethisterone and the
experimental and never-marketed
hormonal antineoplastic agent...
- 17α-Ethenylated/ethynylated
testosterone derivatives:
ethynyltestosterone (
ethisterone) and
vinyltestosterone derivatives The last
group consists of progestins...
-
sometimes designated as
ethinyl in
compounds such as
ethinylestradiol and
ethisterone (ethinyltestosterone). See main page alkynes.
Ethynylation Ethynyl radical...
-
derived from
modification of
ethisterone via
introduction of
methyl groups at the C6α and C21 positions.
Relative to
ethisterone, it is 12 times as potent...
- 17α-Ethynyltestosterone derivatives:
Danazol Gestrinone Progestins (e.g.,
ethisterone (ethynyltestosterone), levonorgestrel, norgestrel,
norethisterone (norethindrone)...
