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Etacstil (developmental code
names GW-5638, DPC974) is an
orally active, nonsteroidal,
combined selective estrogen receptor modulator (SERM) and selective...
- –
Invention of tyrosine-kinase
inhibitor Imatinib 1992 –
Invention of
Etacstil breast cancer anti-estrogen (SERM/SERD)
hormonal therapy drug that overcomes...
- clomifene),
droloxifene (3-hydroxytamoxifen),
etacstil, fispemifene, GW-7604 (4-hydroxyetacstil;
metabolite of
etacstil),
idoxifene (pyrrolidino-4-iodotamoxifen)...
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Cyclofenil D-15413
Desmethylchlorotrianisene Droloxifene Enclomifene Endoxifen Etacstil (GW-5638, DPC-974)
Ethamoxytriphetol (MER-25)
Femarelle Fispemifene GW-7604...
-
Cyclofenil D-15413
Desmethylchlorotrianisene Droloxifene Enclomifene Endoxifen Etacstil (GW-5638, DPC-974)
Ethamoxytriphetol (MER-25)
Femarelle Fispemifene GW-7604...
-
Cyclofenil D-15413
Desmethylchlorotrianisene Droloxifene Enclomifene Endoxifen Etacstil (GW-5638, DPC-974)
Ethamoxytriphetol (MER-25)
Femarelle Fispemifene GW-7604...
-
Deaminohydroxytoremifene 0.82–2.63 0.59–1.22 ? ? SERM
Bazedoxifene – ? ? 0.053 ? SERM
Etacstil GW-5638 4.30 11.5 ? ? SERM ICI-164,384 – 63.5 (3.70–97.7) 166 0.2 0.08...
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Deaminohydroxytoremifene 0.82–2.63 0.59–1.22 ? ? SERM
Bazedoxifene – ? ? 0.053 ? SERM
Etacstil GW-5638 4.30 11.5 ? ? SERM ICI-164,384 – 63.5 (3.70–97.7) 166 0.2 0.08...
-
Cyclofenil D-15413
Desmethylchlorotrianisene Droloxifene Enclomifene Endoxifen Etacstil (GW-5638, DPC-974)
Ethamoxytriphetol (MER-25)
Femarelle Fispemifene GW-7604...
-
Cyclofenil D-15413
Desmethylchlorotrianisene Droloxifene Enclomifene Endoxifen Etacstil (GW-5638, DPC-974)
Ethamoxytriphetol (MER-25)
Femarelle Fispemifene GW-7604...
