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Erteberel (INNTooltip
International Nonproprietary Name,
USANTooltip United States Adopted Name;
former developmental code name LY-500307; also known...
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functional selectivity for the ERβ over the ERα. An
enantiomer of SERBA-2,
erteberel (SERBA-1), is more
potent and
selective in
comparison and is
under development...
- (fenocycline)
Doisynolic acid
Efavirenz Elacestrant ERB-196 (WAY-202196)
Erteberel (SERBA-1, LY-500307)
Estrobin (DBE)
Fenestrel FERb 033
Fosfestrol (diethylstilbestrol...
- (fenocycline)
Doisynolic acid
Efavirenz Elacestrant ERB-196 (WAY-202196)
Erteberel (SERBA-1, LY-500307)
Estrobin (DBE)
Fenestrel FERb 033
Fosfestrol (diethylstilbestrol...
- (fenocycline)
Doisynolic acid
Efavirenz Elacestrant ERB-196 (WAY-202196)
Erteberel (SERBA-1, LY-500307)
Estrobin (DBE)
Fenestrel FERb 033
Fosfestrol (diethylstilbestrol...
-
postmenopausal women and in
individuals of
either ****.
Diarylpropionitrile ERB-196
Erteberel FERb 033
Prinaberel WAY-166818 WAY-214156
Malamas MS,
Manas ES, McDevitt...
- (fenocycline)
Doisynolic acid
Efavirenz Elacestrant ERB-196 (WAY-202196)
Erteberel (SERBA-1, LY-500307)
Estrobin (DBE)
Fenestrel FERb 033
Fosfestrol (diethylstilbestrol...
- 0.27 67–72 ? ? ERβ
agonist ERB-196 WAY-202,196 ? 180 ? ? ERβ
agonist Erteberel SERBA-1; LY-500,307 ? ? 2.68 0.19 ERβ
agonist SERBA-2 – ? ? 14.5 1.54...
- (fenocycline)
Doisynolic acid
Efavirenz Elacestrant ERB-196 (WAY-202196)
Erteberel (SERBA-1, LY-500307)
Estrobin (DBE)
Fenestrel FERb 033
Fosfestrol (diethylstilbestrol...
- (fenocycline)
Doisynolic acid
Efavirenz Elacestrant ERB-196 (WAY-202196)
Erteberel (SERBA-1, LY-500307)
Estrobin (DBE)
Fenestrel FERb 033
Fosfestrol (diethylstilbestrol...