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Gabapentin enacarbil (Horizant (ER) (U.S.Tooltip
United States),
Regnite (in ****an)) is an
anticonvulsant and
analgesic drug of the
gabapentinoid class...
- pregabalin, and mirogabalin, as well as a
gabapentin prodrug,
gabapentin enacarbil.
Further analogues like
imagabalin and
atagabalin have been
tested in...
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Gabapentinoids (α2δ ligands),
including gabapentin, pregabalin, and
gabapentin enacarbil, are also
widely used in the
treatment of RLS. They are used as first-line...
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prodrugs are such as
dabigatran etexilate (approved in 2010),
gabapentin enacarbil (2011),
sofosbuvir (2013),
tedizolid phosphate (2014), isavuconazonium...
- anticonvulsant;
inhibitor of α2δ subunit-containing
VGCCs Gabapentin enacarbil – used for the
treatment of
restless legs
syndrome and
postherpetic neuralgia;...
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tried by
Pfizer as a
treatment for insomnia. A
prodrug form (gabapentin
enacarbil) was
approved by the U.S. Food and Drug
Administration (FDA). When taken...
- S2CID 5349255.
Iftikhar IH,
Alghothani L,
Trotti LM (December 2017). "Gabapentin
enacarbil,
pregabalin and
rotigotine are
equally effective in
restless legs syndrome:...
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Orexin Daridorexant Lemborexant Suvorexant α2δ VDCC
Gabapentin Gabapentin enacarbil Mirogabalin Phenibut Pregabalin Others Cannabidiol Cannabis Chlorophenylalkyldiols...
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Calcium blockers Alcohol (ethanol)
Gabapentin Gabapentin enacarbil Leconotide Mirogabalin Pregabalin Ziconotide Sodium blockers Carbamazepine Lacosamide...
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Calcium blockers Alcohol (ethanol)
Gabapentin Gabapentin enacarbil Leconotide Mirogabalin Pregabalin Ziconotide Sodium blockers Carbamazepine Lacosamide...
