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Norepinephrine transporter 27,000–30,500 (Ki) 360–405 (IC50) 54–110 (EC50) (rat)
DATTooltip Dopamine transporter 6,500–>10,000 (Ki) 1,440–21,000 (IC50) 51–278 (EC50)...
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sites on the
monoamine transporters (SERTTooltip
serotonin transporter,
DATTooltip dopamine transporter,
NETTooltip norepinephrine transporter). It is ****ociated...
- 108 ND
Inhibitor NETTooltip Norepinephrine transporter 36 ND
Inhibitor DATTooltip Dopamine transporter 5489 ND
Inhibitor 5-HT1A 5300 3200
Agonist 5-HT2A...
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transporter 5,000 (IC50Tooltip Half-maximal
inhibitory concentration) Rat
DATTooltip Dopamine transporter 29,000 (IC50) Rat
VDCCTooltip Voltage-dependent calcium...
-
NETTooltip Norepinephrine transporter 5,600–>30,000 (Ki) >100,000 (IC50)
DATTooltip Dopamine transporter >30,000 (Ki) >100,000 (IC50) Notes: The
smaller the...
- v t e
Monoamine reuptake inhibitors DATTooltip Dopamine transporter (DRIsTooltip
Dopamine reuptake inhibitors)
NETTooltip Norepinephrine transporter (NRIsTooltip...
- 23–40 401–484 Rat
NETTooltip Norepinephrine transporter 240+ 340+ Rat
DATTooltip Dopamine transporter 1000+ 1000+ Rat 5-HT1A 1000+ 1000+ Rat 5-HT1B/1D...
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multiple mechanisms. The
language employs three applicative prefixes:
DATTooltip Dative case ko-,
INSTooltip Instrumental case e- , and
LOCTooltip Locative...
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Inhibitor Human NETTooltip Norepinephrine transporter >10,000
Inhibitor Human DATTooltip Dopamine transporter >10,000
Inhibitor Human PCP2 154
agonist Human [3H]5-HT...
-
Human NETTooltip Norepinephrine transporter 82–291 IC50
Inhibitor Human DATTooltip Dopamine transporter 63 Ki
Inhibitor Rat HCN1Tooltip Hyperpolarization-activated...