-
Human NETTooltip Norepinephrine transporter 82–291 IC50
Inhibitor Human DATTooltip Dopamine transporter 63 Ki
Inhibitor Rat HCN1Tooltip Hyperpolarization-activated...
-
Norepinephrine transporter 27,000–30,500 (Ki) 360–405 (IC50) 54–110 (EC50) (rat)
DATTooltip Dopamine transporter 6,500–>10,000 (Ki) 1,440–21,000 (IC50) 51–278 (EC50)...
- v t e
Monoamine reuptake inhibitors DATTooltip Dopamine transporter (DRIsTooltip
Dopamine reuptake inhibitors)
NETTooltip Norepinephrine transporter (NRIsTooltip...
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NETTooltip Norepinephrine transporter 5,600–>30,000 (Ki) >100,000 (IC50)
DATTooltip Dopamine transporter >30,000 (Ki) >100,000 (IC50) Notes: The
smaller the...
- v t e
Monoamine reuptake inhibitors DATTooltip Dopamine transporter (DRIsTooltip
Dopamine reuptake inhibitors)
NETTooltip Norepinephrine transporter (NRIsTooltip...
-
transporter 0.15–3.3
Human NETTooltip Norepinephrine transporter 420–925
Human DATTooltip Dopamine transporter 22–315
Human 5-HT1A >35,000
Human 5-HT2A 2,207 Rat...
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transporter 15.2
Human NETTooltip Norepinephrine transporter 1,440
Human DATTooltip Dopamine transporter 1,060
Human 5-HT2A 3,130 Rat 5-HT2C 3,120 Rat H1...
- 23–40 401–484 Rat
NETTooltip Norepinephrine transporter ≥240 ≥340 Rat
DATTooltip Dopamine transporter >1,000 >1,000 Rat 5-HT1A >1,000 >1,000 Rat 5-HT1B/1D...
- v t e
Monoamine reuptake inhibitors DATTooltip Dopamine transporter (DRIsTooltip
Dopamine reuptake inhibitors)
NETTooltip Norepinephrine transporter (NRIsTooltip...
-
NETTooltip Norepinephrine transporter 13,000 (Ki) 14,000 (IC50) >10,000 (EC50)
DATTooltip Dopamine transporter 6,000–>30,000 (Ki) >100,000 (IC50) >10,000 (EC50)...
