-
Ciproxifan is an
extremely potent histamine H3
inverse agonist/antagonist. The
histamine H3
receptor is an
inhibitory autoreceptor located on histaminergic...
-
Examples of
selective H3-antihistamines include:
Clobenpropit ABT-239
Ciproxifan Conessine A-349,821.
Thioperamide H4-antihistamines
inhibit the activity...
-
Examples of
selective H3
antagonists include clobenpropit, ABT-239,
ciproxifan, conessine, A-349,821, enerisant, betahistine, and pitolisant. The histamine...
-
Betahistine (also weak H1 agonist)
Burimamide (also weak H2 antagonist)
Ciproxifan Clobenpropit (also H4 antagonist)
Conessine Failproxifan[citation needed]...
- A-349821 A-423579 ABT-239 ABT-652 AZD5213
Bavisant Betahistine Burimamide Ciproxifan Clobenpropit Conessine Enerisant GSK-189254
Impentamine Iodophenpropit...
- A-349821 A-423579 ABT-239 ABT-652 AZD5213
Bavisant Betahistine Burimamide Ciproxifan Clobenpropit Conessine Enerisant GSK-189254
Impentamine Iodophenpropit...
- A-349821 A-423579 ABT-239 ABT-652 AZD5213
Bavisant Betahistine Burimamide Ciproxifan Clobenpropit Conessine Enerisant GSK-189254
Impentamine Iodophenpropit...
- A-349821 A-423579 ABT-239 ABT-652 AZD5213
Bavisant Betahistine Burimamide Ciproxifan Clobenpropit Conessine Enerisant GSK-189254
Impentamine Iodophenpropit...
- at the
human H3
receptor than
comparable agents such as thioperamide,
ciproxifan, and cipralisant. It was
ultimately dropped from
human trials after showing...
- A-349821 A-423579 ABT-239 ABT-652 AZD5213
Bavisant Betahistine Burimamide Ciproxifan Clobenpropit Conessine Enerisant GSK-189254
Impentamine Iodophenpropit...
