-
Buspirone, sold
under the
brand name Buspar,
among others, is an anxiolytic, a
medication primarily used to
treat anxiety disorders,
particularly generalized...
- Side
effects of
buspirone by
incidence include: Very
common (>10% incidence) Dizziness/lightheadedness
Headache Somnolence (sleepiness)
Common (1–10%...
-
anxiety disorders due to
their fast
onset but
carry the risk of dependence.
Buspirone is
indicated for GAD,
which has much
slower onset but with the advantage...
- A
number of
pyrimidinylpiperazine derivatives are drugs, including:
Buspirone –
anxiolytic Dasatinib –
anticancer agent Eptapirone –
anxiolytic Gepirone –...
-
Buspirone/testosterone (tentative
brand name Lybridos) is a
combination of
buspirone, a 5-HT1A
receptor partial agonist, α2-adrenergic
receptor antagonist...
- (S-20,499)
Binospirone (MDL-73,005) BMY-7,378 (CAS number: 21102-95-4 )
Buspirone (Buspar)
Enilospirone (CERM-3,726)
Eptapirone (F-11,440)
Gepirone (Exxua)...
- to
moderate cerebellar ataxia may be
treatable with
buspirone. It is
thought that the
buspirone increases the
serotonin levels in the
cerebellum and...
- the D2
receptor (30- to 50-fold
lower in
comparison to
buspirone). However,
similarly to
buspirone,
gepirone metabolizes into 1-(2-pyrimidinyl)piperazine...
-
specific type of receptor. E.g.
buspirone is a
selective agonist for
serotonin 5-HT1A.
Partial agonists (such as
buspirone, aripiprazole, buprenorphine,...
- have been
classed as
partial agonists at
particular receptors include buspirone, aripiprazole, buprenorphine,
nalmefene and norclozapine.
Examples of...
