-
Bosentan, sold
under the
brand name
Tracleer among others, is a dual
endothelin receptor antagonist medication used in the
treatment of
pulmonary artery...
-
which affect both
endothelin A (ETA) and B
receptors (ETB) aprocitentan,
bosentan, macitentan,
tezosentan Selective ETA
Receptor Antagonists,
which affect...
- (COX-2 inhibitor)
Celecoxib (COX-2 inhibitor)
Parecoxib (COX-2 inhibitor)
Bosentan (endothelin
receptor antagonist)
Dofetilide (class III antiarrhythmic)...
-
treat pulmonary hypertension include epoprostenol, treprostinil, iloprost,
bosentan, ambrisentan, macitentan, and sildenafil, tadalafil, selexipag, riociguat...
-
Examples of such
sodium salts are (selection): Bispyribac, bithionol,
bosentan, brequinar, bromfenac, Cefmenoxime, ceftiofur, citicoline, diclofenac,...
-
bornaprolol (INN)
bornelone (INN)
Borofax bortezomib (USAN)
Boruzu Bosatria bosentan (INN)
bosutinib (USAN, INN)
botiacrine (INN)
Botox Boudreaux's Butt Paste...
- high
receptor occupancy half-life (approximately 17 minutes)
compared to
bosentan (approximately 70 seconds) and
ambrisentan (approximately 40 seconds)....
- same as
bosentan, but the
hepatotoxicity of
sitaxentan outweighs its benefits.
Dosing is once daily, as
opposed to
twice daily for
bosentan. On December...
-
hypertension in Raynaud's phenomenon, and the
endothelin receptor antagonist bosentan is used to
manage severe pulmonary hypertension and
prevent finger ulcers...
-
pulmonary hypertension,
which was
treatable in
preliminary research by
bosentan,
sitaxentan or ambrisentan.
Endothelins have
involvement in cardiovascular...
