-
substituted benzothiophenes have been little-encountered as
designer drugs as of 2022.
Tactogen has
patented a
number of
benzothiophenes as
novel entactogens...
-
manufacturing of dyes such as thioindigo. Most
syntheses of
benzothiophene create substituted benzothiophenes as a
precursor to
further reactions. An
example is...
- of 4-hydroxytamoxifen.
Raloxifene belongs to the second-generation
benzothiophene SERM drugs. It has a high
affinity for the ER with
potent antiestrogenic...
-
include metal-free
alkylation and
arylation of
benzothiophenes, metal-free
synthesis of
benzothiophenes by
twofold C–H functionalization, and new reagents...
-
petroleum ranging from
thiophene itself to more
condensed derivatives,
benzothiophenes and dibenzothiophenes.
Thiophene itself and its
alkyl derivatives are...
-
benzothiophene group. It is
closely related to 5-MAPB but with the
oxygen atom
replaced by sulfur,
changing the core ring
structure to
benzothiophene...
- (6-MABB) Dihydrobenzofurans: 5-APDB 5-MAPDB 6-APDB 6-MAPDB IBF5MAP
Benzothiophenes: 5-APBT 5-MAPBT 6-APBT 6-MAPBT Indanes: 5-APDI 5-MAPDI Indoles: 5-IT...
-
Bioisosteres Benzofurans (e.g., 5-MeO-DiBF,
dimemebfe (5-MeO-BFE), mebfap)
Benzothiophenes (e.g., 3-APBT)
Indazoles (e.g., AL-38022A)
Indenes (e.g., C-DMT) Isotryptamines...
- fenfluramine, the
rigid 4-chloro
phenethylamine lorcaserin, and the
benzothiophenes 5-APBT and 6-APBT.
Certain other phenethylamines, like naphthylaminopropane...
-
furans and
benzofurans Asymmetric hydrogenation of
thiophenes and
benzothiophenes has been
catalyzed by some ruthenium(II)
complexes of N-heterocyclic...
