-
release (EC50Tooltip half-maximal
effective concentration, nM) of
arylpiperazines Compound PAL #
Serotonin Norepinephrine Dopamine Type Ref 1-Benzylpiperazine...
-
benzamide N05AL07
Lumateperone Caplyta butyrophenone Lurasidone Latuda n-
arylpiperazine (piperazine) N05AE05
Melperone Bunil, Buronil,
Eunerpan butyrophenone...
- (2): 151–7. PMID 20369792.
Caccia S (August 2007). "N-dealkylation of
arylpiperazine derivatives:
disposition and
metabolism of the 1-aryl-piperazines formed"...
- Amphetamine-type/dopamine
releasing agents:
Alkylamines Cycloalkylaminopropanes Arylpiperazines Benzylpiperazines Phenylpiperazines Phenethylamines Aminorexes/phenyloxazolamines...
- lysergamides: 12-Hydroxy-LSD 12-Methoxy-LSD Bioisosteres: JRT
Others Arylpiperazines (e.g., 2C-B-PP, 2-NP, MK-212, ORG-12962, pCPP, mCPP, pFPP, quipazine...
- Amphetamine-type/dopamine
releasing agents:
Alkylamines Cycloalkylaminopropanes Arylpiperazines Benzylpiperazines Phenylpiperazines Phenethylamines Aminorexes/phenyloxazolamines...
- Amphetamine-type/dopamine
releasing agents:
Alkylamines Cycloalkylaminopropanes Arylpiperazines Benzylpiperazines Phenylpiperazines Phenethylamines Aminorexes/phenyloxazolamines...
-
selective 5-HT1A
receptor partial agonist (Ki = 0.1 nM; IA = 40%) with an
arylpiperazine structure. It is one of the
highest affinity ligands for the 5-HT1A...
- lysergamides: 12-Hydroxy-LSD 12-Methoxy-LSD Bioisosteres: JRT
Others Arylpiperazines (e.g., 2C-B-PP, 2-NP, MK-212, ORG-12962, pCPP, mCPP, pFPP, quipazine...
- Amphetamine-type/dopamine
releasing agents:
Alkylamines Cycloalkylaminopropanes Arylpiperazines Benzylpiperazines Phenylpiperazines Phenethylamines Aminorexes/phenyloxazolamines...
