-
Substituted arylalkylamines are a
group of
chemical compounds.
These compounds are
divided into two main categories:
indolylalkylamines and phenylalkylamines...
-
selectivity for SERT and DAT,
namely the 4-indolyl and 1-naphthyl
arylalkylamines ent-16b (Ki 0.82, 3.8, 4840 nM for SERT, DAT, NET) and ent-13b respectively...
- Weinheim: Wiley-VCH. ISBN 978-3-527-66445-0. Dörwald FZ, ed. (2012). "46.
Arylalkylamines". Lead
optimization for
medicinal chemists:
pharmacokinetic properties...
- Weinheim: Wiley-VCH. ISBN 978-3-527-66445-0. Dörwald FZ, ed. (2012). "46.
Arylalkylamines". Lead
optimization for
medicinal chemists :
pharmacokinetic properties...
- the cAMP-dependent
protein kinase A (PKA). PKA then
phosphorylates arylalkylamine N-acetyltransferase (AANAT), the
penultimate enzyme in the melatonin...
- of
cerebral 5-hydroxytryptamine and 5-hydroxyindolacetic acid by an
arylalkylamine". Life Sciences. 2 (11): 828–833. doi:10.1016/0024-3205(63)90094-8....
-
Aralkylamine N-acetyltransferase (AANAT) (EC 2.3.1.87), also
known as
arylalkylamine N-acetyltransferase or
serotonin N-acetyltransferase (SNAT), is an enzyme...
-
Institute on Drug Abuse: Rockville, MD, 1994.
Glennon RA (October 1999). "
Arylalkylamine drugs of abuse: an
overview of drug
discrimination studies". Pharmacology...
- 1007/BF02245118. PMID 1387963. S2CID 24965789. Dörwald FZ, ed. (2012). "46.
Arylalkylamines". Lead
optimization for
medicinal chemists :
pharmacokinetic properties...
- N-(trifluoroacetyl)-α-amino acid chlorides.
Application to the
preparation of β-
arylalkylamines and 3-substituted 1,2,3,4-tetrahydroisoquinolines." J. Org. Chem. 49...
