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Substituted arylalkylamines are a
group of
chemical compounds.
These compounds are
divided into two main categories:
indolylalkylamines and phenylalkylamines...
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Aralkylamine N-acetyltransferase (AANAT) (EC 2.3.1.87), also
known as
arylalkylamine N-acetyltransferase or
serotonin N-acetyltransferase (SNAT), is an enzyme...
- the cAMP-dependent
protein kinase A (PKA). PKA then
phosphorylates arylalkylamine N-acetyltransferase (AANAT), the
penultimate enzyme in the melatonin...
- Weinheim: Wiley-VCH. ISBN 978-3-527-66445-0. Dörwald FZ, ed. (2012). "46.
Arylalkylamines". Lead
optimization for
medicinal chemists:
pharmacokinetic properties...
- Weinheim: Wiley-VCH. ISBN 978-3-527-66445-0. Dörwald FZ, ed. (2012). "46.
Arylalkylamines". Lead
optimization for
medicinal chemists :
pharmacokinetic properties...
-
Institute on Drug Abuse: Rockville, MD, 1994.
Glennon RA (October 1999). "
Arylalkylamine drugs of abuse: an
overview of drug
discrimination studies". Pharmacology...
- of
cerebral 5-hydroxytryptamine and 5-hydroxyindolacetic acid by an
arylalkylamine". Life Sciences. 2 (11): 828–833. doi:10.1016/0024-3205(63)90094-8....
- }
arylalkylamine +
acetate Thus, the two
substrates of this
enzyme are N-acetylarylalkylamine and H2O,
whereas its two
products are
arylalkylamine and...
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selectivity for SERT and DAT,
namely the 4-indolyl and 1-naphthyl
arylalkylamines ent-16b (Ki 0.82, 3.8, 4840 nM for SERT, DAT, NET) and ent-13b respectively...
-
exists for
melatonin secretion in
vertebrates is the
enzyme AANAT (
arylalkylamine N-acetyltransferase). The
expression of the
AANAT gene is controlled...
