- others. High-dose
antigonadotropin therapy has been
referred to as
medical castration. The best-known and
widely used
antigonadotropins are the gonadotropin-releasing...
- and
antigonadotropins. AR
antagonists work by
directly blocking the
effects of androgens,
while androgen synthesis inhibitors and
antigonadotropins work...
-
inhibitors like 5α-reductase
inhibitors and CYP17A1 inhibitors, and
antigonadotropins like GnRH analogues, estrogens, and progestogens. In addition, it...
- (SERD) fulvestrant,
aromatase inhibitors (AIs) like anastrozole, and
antigonadotropins including androgens/anabolic steroids, progestogens, and GnRH analogues...
- steroids.
Steroidogenesis inhibitors are
analogous in
effect and use to
antigonadotropins (which
specifically inhibit gonadal ****
steroid production), but work...
- used as a progonadotropin, all
approved GnRH
agonists are used as
antigonadotropins. The
clinically used
desensitizing GnRH
agonists are
available in...
-
reserved to
describe AR
antagonists (and
sometimes progestogenic antigonadotropins).
Clascoterone (CB-03-01; Breezula, Winlevi): A pure AR antagonist...
-
androgen production in the
gonads are
known as
antigonadotropins.
Estrogens and
progestogens are
antigonadotropins and
hence are
functional antiandrogens. The...
-
suppress gonadotropin or ****
hormone levels like other,
stronger antigonadotropins do), the drug
prevents the mid-cycle
surge in the
levels of these...
- (GnRH)
analogues such as
leuprorelin and cetrorelix, and/or
other antigonadotropins such as
megestrol acetate and
medroxyprogesterone acetate. Androgen...