-
Afimoxifene, also
known as 4-hydroxytamoxifen (4-OHT) and by its
tentative brand name TamoGel, is a
selective estrogen receptor modulator (SERM) of the...
- respectively,
whereas afimoxifene had 178% and 338% of the
affinity of
estradiol for the ERα and ERβ, respectively. Hence,
afimoxifene showed 25-fold higher...
-
tamoxifen is
metabolized by the CYP2D6
enzyme to
produce endoxifen and
afimoxifene (4-hydroxytamoxifen). Currently,
endoxifen is
approved by
Drugs Controller...
-
afatinib (INN, (USAN)
Afaxin a****ostat (USAN, INN)
afelimomab (INN)
afimoxifene (INN)
aflibercept (USAN, INN))
afloqualone (INN)
afovirsen (INN) AFP-Cide...
- triphenylmethylethylene; the
selective estrogen receptor modulators (SERMs)
afimoxifene, brilanestrant, broparestrol, clomifene, clomifenoxide, droloxifene,...
- 06–16%). 4-Hydroxyclomifene, a
major active metabolite of clomifene, and
afimoxifene (4-hydroxytamoxifen), a
major active metabolite of tamoxifen, show 89–251%...
- (GSK-9089) GSK-4716 (GW-4716) SLU-PP-332 Antagonists: 4-Hydroxytamoxifen (
afimoxifene)
Bisphenol AF
Diethylstilbestrol ERRγTooltip Estrogen-related receptor...
- also
protect it from
deactivation from the SERM 4-hydroxytamoxifen (
afimoxifene). This may be the
mechanism by
which BPA acts as a xenoestrogen. Different...
- 4'-Hydroxynorendoxifen 27-Hydroxycholesterol
Acefluranol Acolbifene Afimoxifene Anordiol Anordrin Arzoxifene Bazedoxifene Brilanestrant Broparestrol...
-
currently under development and in
clinical trials include acolbifene,
afimoxifene (4-hydroxytamoxifen;
metabolite of tamoxifen), elacestrant, enclomifene...
